PF-04981517

CHF 60.00
In stock
SYN-3007-M0011 mgCHF 60.00
SYN-3007-M0055 mgCHF 108.00
SYN-3007-M01010 mgCHF 227.00
SYN-3007-M05050 mgCHF 718.00
SYN-3007-M100100 mgCHF 1'251.00
 
More Information
Product Details
Synonyms CYP3CIDE
Product Type Chemical
Properties
Formula C26H32N8
MW 456.6
CAS 1390637-82-7
Purity Chemicals ≥95%
Appearance Solid.
Solubility Soluble in DMSO. Slightly soluble (<1mg/ml) in ethanol.
Declaration Manufactured by SynKinase.
Other Product Data Target: CYP3A4 - CYP3A4 - CYP3A5 - CYP3A7 | Kinase Group: Pfizer Licensed | Substrate: N/A

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Our product description may differ slightly from the original manufacturers product datasheet.
InChi Key WDWIMDKOXZZYHH-FQEVSTJZSA-N
Shipping and Handling
Shipping AMBIENT
Short Term Storage +4°C
Long Term Storage -20°C
Use/Stability Stable for at least 2 years after receipt when stored at -20°C.
Documents
MSDS Inquire
Product Specification Sheet
Datasheet Download PDF
PF-04981517 is a potent and selective enzyme inhibitor of CYP3A4 with IC(50) values of 0.03, 17 and 70M for CYP3A4, CYP3A5 and CYP3A7, respectively.
Product References
  1. The novel and orally active thrombin receptor antagonist E5555 (Atopaxar) inhibits arterial thrombosis without affecting bleeding time in guinea pigs: M. Kogushi, et al.; Eur. J. Pharmacol. 657, 131 (2011)
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