Cookie Policy: This site uses cookies to improve your experience. You can find out more about our use of cookies in our Privacy Policy. By continuing to browse this site you agree to our use of cookies.
Cayman
ENPP1 Inhibitor 4e
62
CHF
CHF 62.00
In stock
CAY-37687-55 mgCHF 62.00
CAY-37687-2525 mgCHF 168.00
CAY-37687-5050 mgCHF 303.00
| Product Details | |
|---|---|
| Synonyms | cGAMP-compound 4e |
| Product Type | Chemical |
| Properties | |
| Formula | C16H12FN5O2S |
| MW | 357.4 |
| Purity Chemicals | ≥98% |
| Appearance | A solid |
| Declaration | Manufactured by Cayman Chemicals. |
| Other Product Data |
Click here for Original Manufacturer Product Datasheet |
| InChi Key | PTZJKRPYZKMREN-UHFFFAOYSA-N |
| Smiles | FC(C=C1)=CC2=C1C(NC(CSC3=NC4=NC(OC)=CC=C4N3)=N2)=O |
| Shipping and Handling | |
| Shipping | BLUE ICE |
| Long Term Storage | -20°C |
| Documents | |
| MSDS | Inquire |
| Product Specification Sheet | |
| Datasheet |
 Download PDF |
Description
An ENPP1 inhibitor (IC50 = 0.188 µM); inhibits ENPP1 in MDA-MB-231 cells (IC50 = 0.732 µM); selectively cytotoxic to 4T1 murine metastatic breast cancer cells (IC50 = 2.99 µM) over non-cancerous L-02 and 293T cells at 50 µM; increases serum levels of IFN-β in mice when administered at a dose of 0.5 mg/kg in combination with cGAMP.