PIK-75

CHF 60.00
In stock
SYN-1067-M0011 mgCHF 60.00
SYN-1067-M0055 mgCHF 78.00
SYN-1067-M01010 mgCHF 90.00
SYN-1067-M05050 mgCHF 329.00
SYN-1067-M100100 mgCHF 461.00
 
More Information
Product Details
Synonyms PIK75
Product Type Chemical
Properties
Formula C16H14BrN5O4S
MW 452.3
CAS 372196-67-3
Purity Chemicals ≥95%
Appearance Solid.
Solubility Soluble in DMSO. Slightly soluble (<1mg/ml) in ethanol.
Declaration Manufactured by SynKinase.
Other Product Data Target: PI3K | Kinase Group: Lipid Kinase | Substrate: Lipid

Click here for Original Manufacturer Product Datasheet
Our product description may differ slightly from the original manufacturers product datasheet.
InChi Key QTHCAAFKVUWAFI-DJKKODMXSA-N
Shipping and Handling
Shipping AMBIENT
Short Term Storage +4°C
Long Term Storage -20°C
Use/Stability Stable for at least 2 years after receipt when stored at -20°C.
Documents
MSDS Download PDF
Product Specification Sheet
Datasheet Download PDF
PIK-75 is a PI3K inhibitor displaying selectivity for the p110α isoform (IC(50) of 6nM). PIK-75 blocks the phosphorylation of PKB induced by insulin.
Product References
  1. Phosphoinositide-3-kinases (PI3Ks): combined comparative modeling and 3D-QSAR to rationalize the inhibition of p110alpha: R. Frederick & W.A. Denny; J. Chem. Inf. Model 48, 629 (2008)
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