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SynKinase
PIK-294
CHF 0.00
In stock
SYN-1098-M0011 mgCHF 149.00
SYN-1098-M0055 mgCHF 227.00
SYN-1098-M01010 mgCHF 412.00
SYN-1098-M05050 mgCHF 1'263.00
SYN-1098-M100100 mgINQ
Product Details | |
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Synonyms | PIK294 |
Product Type | Chemical |
Properties | |
Formula | C28H23N7O2 |
MW | 489.5 |
CAS | 900185-02-6 |
Purity Chemicals | ≥95% |
Appearance | Solid. |
Solubility | Soluble in DMSO. Slightly soluble (<1mg/ml) in ethanol. |
Declaration | Manufactured by SynKinase. |
Other Product Data |
Target: PI3K | Kinase Group: Lipid Kinase | Substrate: Lipid Click here for Original Manufacturer Product Datasheet Our product description may differ slightly from the original manufacturers product datasheet. |
InChi Key | WFSLJOPRIJSOJR-UHFFFAOYSA-N |
Shipping and Handling | |
Shipping | AMBIENT |
Short Term Storage | +4°C |
Long Term Storage | -20°C |
Use/Stability | Stable for at least 2 years after receipt when stored at -20°C. |
Documents | |
MSDS | Download PDF |
Product Specification Sheet | |
Datasheet | Download PDF |
Description
PIK-294 is a PI3 Kinase inhibitor that is 20- to 60-fold more potent than the parent compound, PIK-293. It is one of the most potent p110δ-selective inhibitors that has been reported, with an IC(50) of 10nM.
Product References
- A pharmacological map of the PI3-K family defines a role for p110alpha in insulin signaling: Z.A. Knight, et al.; Cell 125, 733 (2006)